Pharmacology · Pharmacokinetics and Pharmacodynamics

A patient is receiving vancomycin with an AUC/MIC-guided dosing strategy. The AUC0-24/MIC target for MRSA bacteremia is 400–600 mg·h/L. Compared to trough-only monitoring, AUC/MIC-guided dosing reduces which complication?

  • A Vancomycin-associated nephrotoxicity by preventing unnecessarily high trough concentrations (which correlate with AUC), while maintaining therapeutic AUC/MIC targets
  • B Risk of Clostridium difficile infection by reducing total drug exposure
  • C Risk of ototoxicity by keeping peak concentrations below 35 mg/L
  • D The emergence of vancomycin-resistant Enterococcus through lower cumulative drug exposure
Correct answer: A. Vancomycin-associated nephrotoxicity by preventing unnecessarily high trough concentrations (which correlate with AUC), while maintaining therapeutic AUC/MIC targets

Explanation

Vancomycin nephrotoxicity correlates most strongly with AUC24 (total drug exposure over 24 hours) rather than with peak or trough concentrations alone. Traditional trough-only monitoring (targeting 15–20 mg/L) frequently resulted in excessive AUC values and consequent nephrotoxicity without ensuring therapeutic efficacy. AUC/MIC-guided dosing (target AUC0-24 = 400–600 mg·h/L for MRSA) directly measures the relevant pharmacodynamic target, allowing dose optimization that achieves efficacy (AUC/MIC ≥400) while avoiding nephrotoxicity from excessive AUC exposure. The 2020 ASHP/IDSA/SIDP vancomycin monitoring guidelines endorsed this AUC-guided approach. Ototoxicity with modern vancomycin formulations is rare; VRE emergence is primarily an ecological/antibiotic stewardship issue.

Reference: KD Tripathi, Essentials of Medical Pharmacology, 8th ed.

High-yield for: NEET PGINI-CETNExTFMGEUSMLEPLABMRCP

Written and medically reviewed by the StethoPrep medical team.

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