Pharmacology · Antidiabetic Drugs (Oral Hypoglycemics, Insulins)

A 65-year-old man on metformin 1 g twice daily for 8 years presents with fatigue, glossitis, and bilateral lower limb paresthesia. Blood smear shows macro-ovalocytes with hypersegmented neutrophils. Which mechanism explains this deficiency caused by long-term metformin use?

  • A Metformin inhibits intrinsic factor secretion from parietal cells
  • B Metformin destroys gut flora that synthesize B12
  • C Metformin impairs calcium-dependent B12 absorption in the terminal ileum
  • D Metformin increases renal excretion of vitamin B12
Correct answer: C. Metformin impairs calcium-dependent B12 absorption in the terminal ileum

Explanation

Long-term metformin use causes vitamin C12 deficiency in up to 30% of patients by interfering with the calcium-dependent membrane action required for C12-intrinsic factor complex absorption in the terminal ileum. Supplementing calcium can partially reverse this effect. This can lead to megaloblastic anemia and irreversible peripheral neuropathy if undetected.

Reference: Harrison's Principles of Internal Medicine, 21st ed.

High-yield for: NEET PGINI-CETNExTFMGEUSMLEPLABMRCP

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